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Facile, novel two-step syntheses of benzimidazoles, bis-benzimidazoles, and bis-benzimidazole-dihydroquinoxalines

Three scaffolds of benzimidazoles, bis-benzimidazoles, and bis-benzimidazole-dihydroquinoxalines were synthesized via Ugi/de-protection/cyclization methodology. Benzimidazole forming ring closure was enabled under microwave irradiation in the presence of 10% TFA/DCE. The methodology demonstrates the...

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Autors principals: Xu, Zhigang, Shaw, Arthur Y., Dietrich, Justin, Cappelli, Alexandra P., Nichol, Gary, Hulme, Christopher
Format: Artigo
Idioma:Inglês
Publicat: 2012
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC3311162/
https://ncbi.nlm.nih.gov/pubmed/22237832
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1007/s11030-011-9354-x
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