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Pharmacokinetics and Pharmacodynamics of TMC207 and Its N-Desmethyl Metabolite in a Murine Model of Tuberculosis

TMC207 is a first-in-class diarylquinoline with a new mode of action against mycobacteria targeting the ATP synthase. It is metabolized to an active derivative, N-desmethyl TMC207, and both compounds are eliminated with long terminal half-lives (50 to 60 h in mice) reflecting slow release from tissu...

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Autors principals: Rouan, Marie-Claude, Lounis, Nacer, Gevers, Tom, Dillen, Lieve, Gilissen, Ron, Raoof, Araz, Andries, Koen
Format: Artigo
Idioma:Inglês
Publicat: American Society for Microbiology 2012
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC3294950/
https://ncbi.nlm.nih.gov/pubmed/22155815
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1128/AAC.00720-11
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