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Equilibrium binding of carcinogens and antitumor antibiotics to DNA: site selectivity, cooperativity, allosterism.

The equilibrium binding of the carcinogens N-hydroxy-N-acetyl-2-amino-fluorene (HAAF) and 4-nitroquinoline-1-oxide (NQO) to phi X174RF DNA have been studied by phase partition techniques. Both molecules bind in a cooperative manner with only a few carcinogen molecules binding to each phi X174RF DNA...

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Detalhes bibliográficos
Publicado no:Nucleic Acids Res
Main Authors: Winkle, S A, Krugh, T R
Formato: Artigo
Idioma:Inglês
Publicado em: Oxford University Press 1981
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.govhttps://pmc.ncbi.nlm.nih.gov/articles/PMC327340/
https://ncbi.nlm.nih.govhttps://pubmed.ncbi.nlm.nih.gov/6456451/
https://ncbi.nlm.nih.govhttps://doi.org/10.1093/nar/9.13.3175
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