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Rationalizing Tight Ligand Binding through Cooperative Interaction Networks

[Image: see text] Small modifications of the molecular structure of a ligand sometimes cause strong gains in binding affinity to a protein target, rendering a weakly active chemical series suddenly attractive for further optimization. Our goal in this study is to better rationalize and predict the o...

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Autores principales: Kuhn, Bernd, Fuchs, Julian E., Reutlinger, Michael, Stahl, Martin, Taylor, Neil R.
Formato: Artigo
Lenguaje:Inglês
Publicado: American Chemical Society 2011
Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC3246350/
https://ncbi.nlm.nih.gov/pubmed/22087588
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/ci200319e
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