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Discovery of Novel Checkpoint Kinase 1 Inhibitors by Virtual Screening Based on Multiple Crystal Structures

Incorporating receptor flexibility is considered crucial for improvement of docking-based virtual screening. With an abundance of crystallographic structures freely available, docking with multiple crystal structures is believed to be a practical approach to cope with protein flexibility. Here we de...

Deskribapen osoa

Gorde:
Xehetasun bibliografikoak
Egile Nagusiak: Li, Yan, Kim, Dong Joon, Ma, Weiya, Lubet, Ronald A., Bode, Ann M., Dong, Zigang
Formatua: Artigo
Hizkuntza:Inglês
Argitaratua: 2011
Gaiak:
Sarrera elektronikoa:https://ncbi.nlm.nih.gov/pmc/articles/PMC3244973/
https://ncbi.nlm.nih.gov/pubmed/21955044
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/ci200257b
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