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The Discovery of Aurora Kinase Inhibitor by Multi-Docking-Based Virtual Screening

We report the discovery of aurora kinase inhibitor using the fragment-based virtual screening by multi-docking strategy. Among a number of fragments collected from eMololecules, we found four fragment molecules showing potent activity (>50% at 100 μM) against aurora kinase. Based on the explored...

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Publicat a:Int J Mol Sci
Autors principals: Kim, Jun-Tae, Jung, Seo Hee, Kang, Sun Young, Ryu, Chung-Kyu, Kang, Nam Sook
Format: Artigo
Idioma:Inglês
Publicat: MDPI 2014
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC4264174/
https://ncbi.nlm.nih.gov/pubmed/25383681
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/ijms151120403
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