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Targeting Acetylcholinesterase: Identification of Chemical Leads by High Throughput Screening, Structure Determination and Molecular Modeling

Acetylcholinesterase (AChE) is an essential enzyme that terminates cholinergic transmission by rapid hydrolysis of the neurotransmitter acetylcholine. Compounds inhibiting this enzyme can be used (inter alia) to treat cholinergic deficiencies (e.g. in Alzheimer's disease), but may also act as d...

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Detaylı Bibliyografya
Asıl Yazarlar: Berg, Lotta, Andersson, C. David, Artursson, Elisabet, Hörnberg, Andreas, Tunemalm, Anna-Karin, Linusson, Anna, Ekström, Fredrik
Materyal Türü: Artigo
Dil:Inglês
Baskı/Yayın Bilgisi: Public Library of Science 2011
Konular:
Online Erişim:https://ncbi.nlm.nih.gov/pmc/articles/PMC3227566/
https://ncbi.nlm.nih.gov/pubmed/22140425
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1371/journal.pone.0026039
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