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Identification of a GPER/GPR30 Antagonist with Improved Estrogen Receptor Counterselectivity
GPER/GPR30 is a seven-transmembrane G protein-coupled estrogen receptor that regulates many aspects of mammalian biology and physiology. We have previously described both a GPER-selective agonist G-1 and antagonist G15 based on a tetrahydro-3H-cyclopenta[c]quinoline scaffold. The antagonist lacks an...
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| Main Authors: | , , , , , , , , , , , , |
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| Format: | Artigo |
| Jezik: | Inglês |
| Izdano: |
2011
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| Teme: | |
| Online dostop: | https://ncbi.nlm.nih.gov/pmc/articles/PMC3220788/ https://ncbi.nlm.nih.gov/pubmed/21782022 https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.jsbmb.2011.07.002 |
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