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Synthesis and SAR optimization of diketo acid pharmacophore for HCV NS5B polymerase inhibition

Hepatitis C virus (HCV) NS5B polymerase is a key target for anti-HCV therapeutics development. Here we report the synthesis and biological evaluation of a new series of α,γ-diketo acids (DKAs) as NS5B polymerase inhibitors. We initiated structure-activity relationship (SAR) optimization around the f...

Deskribapen osoa

Gorde:
Xehetasun bibliografikoak
Egile Nagusiak: Bhatt, Aaditya, Gurukumar, K. R., Basu, Amartya, Patel, Maulik R., Kaushik-Basu, Neerja, Talele, Tanaji T.
Formatua: Artigo
Hizkuntza:Inglês
Argitaratua: 2011
Gaiak:
Sarrera elektronikoa:https://ncbi.nlm.nih.gov/pmc/articles/PMC3208381/
https://ncbi.nlm.nih.gov/pubmed/21893371
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.ejmech.2011.08.028
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