Caricamento...

An NMR strategy for fragment-based ligand screening utilizing a paramagnetic lanthanide probe

A nuclear magnetic resonance-based ligand screening strategy utilizing a paramagnetic lanthanide probe is presented. By fixing a paramagnetic lanthanide ion to a target protein, a pseudo-contact shift (PCS) and a paramagnetic relaxation enhancement (PRE) can be observed for both the target protein a...

Descrizione completa

Salvato in:
Dettagli Bibliografici
Autori principali: Saio, Tomohide, Ogura, Kenji, Shimizu, Kazumi, Yokochi, Masashi, Burke, Terrence R., Inagaki, Fuyuhiko
Natura: Artigo
Lingua:Inglês
Pubblicazione: Springer Netherlands 2011
Soggetti:
Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC3193990/
https://ncbi.nlm.nih.gov/pubmed/21927934
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1007/s10858-011-9566-5
Tags: Aggiungi Tag
Nessun Tag, puoi essere il primo ad aggiungerne! !