Cargando...

Steroidal Bivalent Ligands for the Estrogen Receptor: Design, Synthesis, Characterization and Binding Affinities

Steroidal bivalent ligands for the estrogen receptor (ER) were designed using crystal structures of ERα dimers as a template. The syntheses of several 17α-ethynylestradiol-based bivalent ligands with varying linker compositions and lengths are described. The binding affinities of these bivalent liga...

Descrición completa

Gardado en:
Detalles Bibliográficos
Main Authors: LaFrate, Andrew L., Carlson, Kathryn E., Katzenellenbogen, John A.
Formato: Artigo
Idioma:Inglês
Publicado: 2009
Assuntos:
Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC3178464/
https://ncbi.nlm.nih.gov/pubmed/19394231
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmc.2009.04.016
Tags: Engadir etiqueta
Sen Etiquetas, Sexa o primeiro en etiquetar este rexistro!