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Design, synthesis and initial biological evaluation of a novel pladienolide analog scaffold()

A novel and simplified synthetic scaffold based on pladienolide was designed using a consensus pharmacophore hypothesis. An initial target was synthesized and evaluated to examine the role of the 3-hydroxy group and the methyl groups present at positions 10, 16, 20, 22 in 1, on biological activity....

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Bibliografische gegevens
Hoofdauteurs: Gundluru, Mahesh Kumar, Pourpak, Alan, Cui, Xiaoli, Morris, Stephan W., Webb, Thomas R.
Formaat: Artigo
Taal:Inglês
Gepubliceerd in: 2011
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Online toegang:https://ncbi.nlm.nih.gov/pmc/articles/PMC3171832/
https://ncbi.nlm.nih.gov/pubmed/21927710
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1039/C1MD00040C
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