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Thermodynamics-based drug design: strategies for inhibiting protein–protein interactions

The inhibition of protein–protein interactions and their ensuing signaling processes play an increasingly important role in modern medicine. Small molecular-weight inhibitors that can be administered orally are the preferred approach but efficient strategies for developing them are not yet generally...

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Autori principali: Schön, Arne, Lam, Sonia Y, Freire, Ernesto
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2011
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC3164996/
https://ncbi.nlm.nih.gov/pubmed/21806377
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.4155/fmc.11.81
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