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Sudemycins, novel small molecule analogues of FR901464, induce alternative gene splicing

Two unrelated bacterial natural products, FR901464 and pladienolide B, have previously been shown to have significant anti-tumor activity in vivo. These compounds target the SF3b subunit of the spliceosome, with a derivative of pladienolide (E7107) entering clinical trials for cancer. However, due t...

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Библиографические подробности
Главные авторы: Fan, Liying, Lagisetti, Chandraiah, Edwards, Carol C., Webb, Thomas R., Potter, Philip M.
Формат: Artigo
Язык:Inglês
Опубликовано: 2011
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Online-ссылка:https://ncbi.nlm.nih.gov/pmc/articles/PMC3113647/
https://ncbi.nlm.nih.gov/pubmed/21344922
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/cb100356k
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