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Pharmacokinetics and Pharmacodynamics of TBR-652, a Novel CCR5 Antagonist, in HIV-1-Infected, Antiretroviral Treatment-Experienced, CCR5 Antagonist-Naïve Patients

TBR-652 is a novel CCR5 antagonist with potent in vitro anti-HIV activity. The objective of this study was to determine the pharmacokinetics (PK) and pharmacodynamics (PD) of TBR-652 in HIV-1-infected, antiretroviral treatment-experienced, CCR5 antagonist-naïve patients. A double-blind, placebo-cont...

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Detalhes bibliográficos
Main Authors: Marier, Jean-Francois, Trinh, MyMy, Pheng, Leng Hong, Palleja, Sandra M., Martin, David E.
Formato: Artigo
Idioma:Inglês
Publicado em: American Society for Microbiology 2011
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC3101382/
https://ncbi.nlm.nih.gov/pubmed/21486960
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1128/AAC.00713-10
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