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Metabolic Intermediate Complex Formation of Human Cytochrome P450 3A4 by Lapatinib

Lapatinib, an oral breast cancer drug, has recently been reported to be a mechanism-based inactivator of cytochrome P450 (P450) 3A4 and also an idiosyncratic hepatotoxicant. It was suggested that formation of a reactive quinoneimine metabolite was involved in mechanism-based inactivation (MBI) and/o...

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Detalhes bibliográficos
Main Authors: Takakusa, Hideo, Wahlin, Michelle D., Zhao, Chunsheng, Hanson, Kelsey L., New, Lee Sun, Chan, Eric Chun Yong, Nelson, Sidney D.
Formato: Artigo
Idioma:Inglês
Publicado em: The American Society for Pharmacology and Experimental Therapeutics 2011
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC3100900/
https://ncbi.nlm.nih.gov/pubmed/21363997
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/dmd.110.037531
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