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N,N′-Alkane-diyl-bis-3-picoliniums as Nicotinic Receptor Antagonists: Inhibition of Nicotine-induced Dopamine Release and Hyperactivity
The current study evaluated a new series of N,N′-alkane-diyl-bis-3-picolinium (bAPi) analogs with C(6)–C(12) methylene linkers as nicotinic receptor (nAChR) antagonists, for nicotine-evoked [(3)H]dopamine (DA) overflow, for blood-brain barrier choline transporter affinity and for attenuation of disc...
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| Autori principali: | , , , , , , , , , , , , |
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| Natura: | Artigo |
| Lingua: | Inglês |
| Pubblicazione: |
2008
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| Soggetti: | |
| Accesso online: | https://ncbi.nlm.nih.gov/pmc/articles/PMC3089982/ https://ncbi.nlm.nih.gov/pubmed/18460644 https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/jpet.108.136630 |
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