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Nortriptyline Reverses Corticosteroid Insensitivity by Inhibition of Phosphoinositide-3-Kinase-δ

Corticosteroid insensitivity represents a major barrier to the treatment of chronic obstructive pulmonary disease (COPD) and severe asthma. It is caused by oxidative stress, leading to reduced histone deacetylase-2 (HDAC2) function through activation of phosphoinositide-3-kinase-δ (PI3Kδ). The tricy...

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Autori principali: Mercado, Nicolas, To, Yasuo, Ito, Kazuhiro, Barnes, Peter J.
Natura: Artigo
Lingua:Inglês
Pubblicazione: The American Society for Pharmacology and Experimental Therapeutics 2011
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC3083104/
https://ncbi.nlm.nih.gov/pubmed/21300705
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/jpet.110.175950
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