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Capitalizing on Tumor genotyping: Towards the design of mutation specific inhibitors of Phosphoinsitide-3-Kinase

Phosphatidylinositide-3-kinases (PI3K) PI3Kα, is a lipid kinase frequently mutated in several cancer types. Under normal physiological conditions it initiates a number of signaling pathways by recruiting other kinases, such as Akt, to the plasma membrane. The mutations observed in tumors increase PI...

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Detalhes bibliográficos
Main Authors: Gabelli, Sandra B., Duong-Ly, Krisna, Brower, Evan T., Amzel, L. Mario
Formato: Artigo
Idioma:Inglês
Publicado em: 2010
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC3079044/
https://ncbi.nlm.nih.gov/pubmed/21035489
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.advenzreg.2010.09.013
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