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A Novel Approach for Predicting P-glycoprotein (ABCB1) Inhibition Using Molecular Interaction Fields

P-glycoprotein (Pgp or ABCB1) is an ABC transporter protein involved in intestinal absorption, drug metabolism and brain penetration, and its inhibition can seriously alter a drug's bioavailability and safety. In addition, inhibitors of Pgp can be used to overcome multidrug resistance. Given th...

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Detalhes bibliográficos
Main Authors: Broccatelli, Fabio, Carosati, Emanuele, Neri, Annalisa, Frosini, Maria, Goracci, Laura, Oprea, Tudor I., Cruciani, Gabriele
Formato: Artigo
Idioma:Inglês
Publicado em: 2011
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC3069647/
https://ncbi.nlm.nih.gov/pubmed/21341745
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jm101421d
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