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Ligand Promiscuity between the Efflux Pumps Human P-Glycoprotein and S. aureus NorA

[Image: see text] Thirty-two diverse compounds were evaluated for their ability to inhibit both Pgp-mediated efflux in mouse T-lymphoma L5178 MDR1 and NorA-mediated efflux in S. aureus SA-1199B. Only four compounds were strong inhibitors of both efflux pumps. Three compounds were found to inhibit Pg...

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Bibliografiske detaljer
Main Authors: Brincat, Jean Pierre, Broccatelli, Fabio, Sabatini, Stefano, Frosini, Maria, Neri, Annalisa, Kaatz, Glenn W., Cruciani, Gabriele, Carosati, Emanuele
Format: Artigo
Sprog:Inglês
Udgivet: American Chemical Society 2012
Online adgang:https://ncbi.nlm.nih.gov/pmc/articles/PMC4025771/
https://ncbi.nlm.nih.gov/pubmed/24900460
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/ml200293c
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