A carregar...

Clozapine and other competitive antagonists reactivate risperidone-inactivated h5-HT(7) receptors: radioligand binding and functional evidence for GPCR homodimer protomer interactions

RATIONALE: The h5-HT(7) receptor is subject to inactivation by risperidone and 9-OH-risperidone, apparently through a pseudo-irreversible complex formed between these drugs and the receptor. Although risperidone and 9-OH-risperidone (“inactivating antagonists”) completely inactivate the receptor, on...

ver descrição completa

Na minha lista:
Detalhes bibliográficos
Main Authors: Teitler, Milt, Toohey, Nicole, Knight, Jessica A., Klein, Michael T., Smith, Carol
Formato: Artigo
Idioma:Inglês
Publicado em: 2010
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC3052287/
https://ncbi.nlm.nih.gov/pubmed/20827463
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1007/s00213-010-2001-x
Tags: Adicionar Tag
Sem tags, seja o primeiro a adicionar uma tag!