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Broad Spectrum Antibiotic Activity of the Arylomycin Natural Products is Masked by Natural Target Mutations

Novel classes of broad-spectrum antibiotics are needed to treat multidrug resistant pathogens. The arylomycin class of natural products inhibits a promising antimicrobial target, type I signal peptidase (SPase), but upon initial characterization appeared to lack whole cell activity against most path...

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Autores principales: Smith, Peter A., Roberts, Tucker C., Romesberg, Floyd E.
Formato: Artigo
Lenguaje:Inglês
Publicado: 2010
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC3003444/
https://ncbi.nlm.nih.gov/pubmed/21095572
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.chembiol.2010.09.009
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