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Targeting TORC2 in multiple myeloma with a new mTOR kinase inhibitor

Although preclinical work with rapalogs suggests potential in treatment of multiple myeloma (MM), they have been less successful clinically. These drugs allostearically inhibit the mammalian target of rapamycin kinase primarily curtailing activity of the target of rapamycin complex (TORC)1. To asses...

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Autori principali: Hoang, Bao, Frost, Patrick, Shi, Yijiang, Belanger, Eileen, Benavides, Angelica, Pezeshkpour, Gholam, Cappia, Susanna, Guglielmelli, Tommasina, Gera, Joseph, Lichtenstein, Alan
Natura: Artigo
Lingua:Inglês
Pubblicazione: American Society of Hematology 2010
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC2996116/
https://ncbi.nlm.nih.gov/pubmed/20686120
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1182/blood-2010-05-285726
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