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Selective inhibition of histone deacetylase 6 (HDAC6) induces DNA damage and sensitizes transformed cells to anticancer agents

Histone deacetylase 6 (HDAC6) is structurally and functionally unique among the 11 human zinc-dependent histone deacetylases. Here we show that chemical inhibition with the HDAC6-selective inhibitor tubacin significantly enhances cell death induced by the topoisomerase II inhibitors etoposide and do...

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Autores principales: Namdar, Mandana, Perez, Gisela, Ngo, Lang, Marks, Paul A.
Formato: Artigo
Lenguaje:Inglês
Publicado: National Academy of Sciences 2010
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC2993347/
https://ncbi.nlm.nih.gov/pubmed/21037108
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1073/pnas.1013754107
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