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Human Blood Concentrations of Cotinine, a Biomonitoring Marker for Tobacco Smoke, Extrapolated from Nicotine Metabolism in Rats and Humans and Physiologically Based Pharmacokinetic Modeling

The present study defined a simplified physiologically based pharmacokinetic (PBPK) model for nicotine and its primary metabolite cotinine in humans, based on metabolic parameters determined in vitro using relevant liver microsomes, coefficients derived in silico, physiological parameters derived fr...

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Autori principali: Yamazaki, Hiroshi, Horiuchi, Kana, Takano, Ryohji, Nagano, Taku, Shimizu, Makiko, Kitajima, Masato, Murayama, Norie, Shono, Fumiaki
Natura: Artigo
Lingua:Inglês
Pubblicazione: Molecular Diversity Preservation International (MDPI) 2010
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC2954553/
https://ncbi.nlm.nih.gov/pubmed/20948932
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/ijerph7093406
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