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Human Blood Concentrations of Cotinine, a Biomonitoring Marker for Tobacco Smoke, Extrapolated from Nicotine Metabolism in Rats and Humans and Physiologically Based Pharmacokinetic Modeling

The present study defined a simplified physiologically based pharmacokinetic (PBPK) model for nicotine and its primary metabolite cotinine in humans, based on metabolic parameters determined in vitro using relevant liver microsomes, coefficients derived in silico, physiological parameters derived fr...

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Detalhes bibliográficos
Main Authors: Yamazaki, Hiroshi, Horiuchi, Kana, Takano, Ryohji, Nagano, Taku, Shimizu, Makiko, Kitajima, Masato, Murayama, Norie, Shono, Fumiaki
Formato: Artigo
Idioma:Inglês
Publicado em: Molecular Diversity Preservation International (MDPI) 2010
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC2954553/
https://ncbi.nlm.nih.gov/pubmed/20948932
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/ijerph7093406
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