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Substrate-specific modulation of CYP3A4 activity by genetic variants of cytochrome P450 oxidoreductase (POR)

OBJECTIVES: CYP3A4 receives electrons from P450 oxidoreductase (POR) to metabolize about 50% of clinically used drugs. There is substantial inter-individual variation in CYP3A4 catalytic activity that is not explained by CYP3A4 genetic variants. CYP3A4 is flexible and distensible, permitting it to a...

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Detalhes bibliográficos
Main Authors: Agrawal, Vishal, Choi, Ji Ha, Giacomini, Kathleen M., Miller, Walter L.
Formato: Artigo
Idioma:Inglês
Publicado em: 2010
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC2940949/
https://ncbi.nlm.nih.gov/pubmed/20697309
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1097/FPC.0b013e32833e0cb5
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