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(86)Rb(+) Efflux Mediated by α4β2*-Nicotinic Acetylcholine Receptors with High and Low Sensitivity to Stimulation by Acetylcholine Display Similar Agonist-Induced Desensitization

The nicotinic acetylcholine receptors (nAChR) assembled from α4 and β2 subunits are the most densely expressed subtype in the brain. Concentration-effect curves for agonist activation of α4β2*-nAChR are biphasic. This biphasic agonist sensitivity is ascribed to differences in subunit stoichiometry....

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Bibliografiske detaljer
Main Authors: Marks, Michael J., Meinerz, Natalie M., Brown, Robert W. B., Collins, Allan C.
Format: Artigo
Sprog:Inglês
Udgivet: 2010
Fag:
Online adgang:https://ncbi.nlm.nih.gov/pmc/articles/PMC2935307/
https://ncbi.nlm.nih.gov/pubmed/20599770
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bcp.2010.06.040
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