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Gene Targeting Demonstrates That α4 Nicotinic Acetylcholine Receptor Subunits Contribute to Expression of Diverse [(3)H]Epibatidine Binding Sites and Components of Biphasic (86)Rb(+) Efflux With High and Low Sensitivity to Stimulation by Acetylcholine

[(3)H]Epibatidine binds to nAChR subtypes in mouse brain with higher (K(D)≈0.02 nM) and lower affinity (KD≈7 nM), which can be further subdivided through inhibition by selected agonists and antagonists. These subsets are differentially affected by targeted deletion of α7, β2 or β4 subunits. Most, bu...

Ausführliche Beschreibung

Gespeichert in:
Bibliographische Detailangaben
Hauptverfasser: Marks, Michael J., Meinerz, Natalie M., Drago, John, Collins, Allan C.
Format: Artigo
Sprache:Inglês
Veröffentlicht: 2007
Schlagworte:
Online Zugang:https://ncbi.nlm.nih.gov/pmc/articles/PMC2577786/
https://ncbi.nlm.nih.gov/pubmed/17631923
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.neuropharm.2007.05.021
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