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Epibatidine Binds to Four Sites on the Torpedo Nicotinic Acetylcholine Receptor

The nicotinic acetylcholine receptor (nAChR) from Torpedo electric organ is a pentamer of homologous subunits. This receptor is generally thought to carry two high affinity sites for agonists under equilibrium conditions. Here we demonstrate directly that each Torpedo nAChR carries at least four bin...

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Autori principali: Kawai, Hideki, Dunn, Susan M. J., Raftery, Michael A.
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2007
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC2536623/
https://ncbi.nlm.nih.gov/pubmed/18083118
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bbrc.2007.12.044
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