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Nicotinic Acetylcholine Receptor Accessory Subunits Determine the Activity Profile of Epibatidine Derivatives

Epibatidine is a potent analgetic agent with very high affinity for brain nicotinic acetylcholine receptors (nAChR). We determined the activity profiles of three epibatidine derivatives, RTI-36, RTI-76, and RTI-102, which have affinity for brain nAChR equivalent to that of epibatidine but reduced an...

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Dettagli Bibliografici
Pubblicato in:Mol Pharmacol
Autori principali: Corrie, Lu Wenchi, Stokes, Clare, Wilkerson, Jenny L., Carroll, F. Ivy, McMahon, Lance R., Papke, Roger L.
Natura: Artigo
Lingua:Inglês
Pubblicazione: The American Society for Pharmacology and Experimental Therapeutics 2020
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC7485586/
https://ncbi.nlm.nih.gov/pubmed/32690626
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/molpharm.120.000037
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