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β-lactamase inhibitors display anti-seizure properties in an invertebrate assay

Antibiotics containing a β-lactam ring (e.g., ceftriaxone) display anti-glutamate effects that underlie their efficacy in animal models of CNS diseases (Rothstein et al., 2005). We hypothesized that the structurally related β-lactamase inhibitors (clavulanic acid, tazobactam)- which also contain a β...

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Autores principales: Rawls, Scott M., Karaca, Fatma, Madhani, Isha, Bhojani, Vineeta, Martinez, Rogelilo L., Abou-Gharbia, Magid, Raffa, Robert B.
Formato: Artigo
Lenguaje:Inglês
Publicado: 2010
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC2924441/
https://ncbi.nlm.nih.gov/pubmed/20600649
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.neuroscience.2010.06.041
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