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Synthesis and screening of a CaaL peptide library versus FTase reveals a surprising number of substrates

Proteins bearing a CaaL sequence are typically geranylgeranylated to enable their proper localization and function. We found that many of the dansyl-GCaaL peptides representing mammalian CaaL proteins can be farnesylated by FTase. This result may have important implications for prenylated protein bi...

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Autors principals: Krzysiak, Amanda J., Aditya, Animesh V., Hougland, James L., Fierke, Carol A., Gibbs, Richard A.
Format: Artigo
Idioma:Inglês
Publicat: 2009
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC2922960/
https://ncbi.nlm.nih.gov/pubmed/20005705
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmcl.2009.11.011
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