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Strategies for discovering and derisking covalent, irreversible enzyme inhibitors

This article presents several covalent inhibitors, including examples of successful drugs, as well as highly selective, irreversible inhibitors of emerging therapeutic targets, such as fatty acid amide hydolase. Covalent inhibitors have many desirable features, including increased biochemical effici...

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Detalhes bibliográficos
Main Authors: Johnson, Douglas S, Weerapana, Eranthie, Cravatt, Benjamin F
Formato: Artigo
Idioma:Inglês
Publicado em: 2010
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC2904065/
https://ncbi.nlm.nih.gov/pubmed/20640225
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