Lanean...

Design, Synthesis, and Biological Evaluation of Resveratrol Analogues as Aromatase and Quinone Reductase 2 Inhibitors for Chemoprevention of Cancer

A series of new resveratrol analogues were designed and synthesized and their inhibitory activities against aromatase were evaluated. The crystal structure of human aromatase (PDB 3eqm) was used to rationalize the mechanism of action of the aromatase inhibitor 32 (IC(50) 0.59 µM) through docking, mo...

Deskribapen osoa

Gorde:
Xehetasun bibliografikoak
Egile Nagusiak: Sun, Bin, Hoshino, Juma, Jermihov, Katie, Marler, Laura, Pezzuto, John M., Mesecar, Andrew D., Cushman, Mark
Formatua: Artigo
Hizkuntza:Inglês
Argitaratua: 2010
Gaiak:
Sarrera elektronikoa:https://ncbi.nlm.nih.gov/pmc/articles/PMC2903642/
https://ncbi.nlm.nih.gov/pubmed/20558073
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmc.2010.05.042
Etiketak: Etiketa erantsi
Etiketarik gabe, Izan zaitez lehena erregistro honi etiketa jartzen!