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Design, Synthesis, and Biological Evaluation of Resveratrol Analogues as Aromatase and Quinone Reductase 2 Inhibitors for Chemoprevention of Cancer

A series of new resveratrol analogues were designed and synthesized and their inhibitory activities against aromatase were evaluated. The crystal structure of human aromatase (PDB 3eqm) was used to rationalize the mechanism of action of the aromatase inhibitor 32 (IC(50) 0.59 µM) through docking, mo...

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Detalhes bibliográficos
Main Authors: Sun, Bin, Hoshino, Juma, Jermihov, Katie, Marler, Laura, Pezzuto, John M., Mesecar, Andrew D., Cushman, Mark
Formato: Artigo
Idioma:Inglês
Publicado em: 2010
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC2903642/
https://ncbi.nlm.nih.gov/pubmed/20558073
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmc.2010.05.042
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