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Targeted polypharmacology: Discovery of dual inhibitors of tyrosine and phosphoinositide kinases

The clinical success of multitargeted kinase inhibitors has stimulated efforts to identify promiscuous drugs with optimal selectivity profiles. It remains unclear to what extent such drugs can be rationally designed, particularly for combinations of targets that are structurally divergent. Here we r...

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Autors principals: Apsel, Beth, Blair, Jimmy A., Gonzalez, Beatriz Z., Nazif, Tamim M., Feldman, Morri E., Aizenstein, Brian, Hoffman, Randy, Williams, Roger L., Shokat, Kevan M., Knight, Zachary A.
Format: Artigo
Idioma:Inglês
Publicat: 2008
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC2880455/
https://ncbi.nlm.nih.gov/pubmed/18849971
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/nchembio.117
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