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Seven Transmembrane Receptors as Shapeshifting Proteins: The Impact of Allosteric Modulation and Functional Selectivity on New Drug Discovery

It is useful to consider seven transmembrane receptors (7TMRs) as disordered proteins able to allosterically respond to a number of binding partners. Considering 7TMRs as allosteric systems, affinity and efficacy can be thought of in terms of energy flow between a modulator, conduit (the receptor pr...

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Detalhes bibliográficos
Main Authors: Kenakin, Terry, Miller, Laurence J.
Formato: Artigo
Idioma:Inglês
Publicado em: The American Society for Pharmacology and Experimental Therapeutics 2010
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC2879912/
https://ncbi.nlm.nih.gov/pubmed/20392808
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/pr.108.000992
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