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Impact of Allosteric Modulation in Drug Discovery: Innovation in Emerging Chemical Modalities

[Image: see text] Recent years have seen an unprecedented level of innovation in allosteric drug discovery and development, with multiple drug candidates advancing into clinical studies. From early examples of allosteric drugs like GABA(A) receptor modulators (benzodiazepines) in the 1960s to more r...

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Pubblicato in:ACS Med Chem Lett
Autori principali: Han, Bingsong, Salituro, Francesco G., Blanco, Maria-Jesus
Natura: Artigo
Lingua:Inglês
Pubblicazione: American Chemical Society 2020
Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC7549105/
https://ncbi.nlm.nih.gov/pubmed/33062158
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acsmedchemlett.9b00655
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