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Thiazole, Oxadiazole, and Carboxamide Derivatives of Artemisinin are Highly Selective and Potent Inhibitors of Toxoplasma gondii

We have prepared 23 new dehydroartemisinin (DART) trioxane derivatives (11 thiazoles, 2 oxadiazoles, and 10 carboxamides) and have screened them for in vitro activity in the Toxoplasma lytic cycle. Fifteen (65%) of the derivatives were non-cytotoxic to host cells (TD(50) ≥ 320 μM). Eight thiazole de...

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Bibliografiske detaljer
Main Authors: Hencken, Christopher P., Jones-Brando, Lorraine, Bordón, Claudia, Stohler, Remo, Mott, Bryan T., Yolken, Robert, Posner, Gary H., Woodard, Lauren E.
Format: Artigo
Sprog:Inglês
Udgivet: 2010
Fag:
Online adgang:https://ncbi.nlm.nih.gov/pmc/articles/PMC2865576/
https://ncbi.nlm.nih.gov/pubmed/20373807
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jm901857d
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