Carregant...

Lobelane Inhibits Methamphetamine-Evoked Dopamine Release via Inhibition of the Vesicular Monoamine Transporter-2

Lobeline is currently being evaluated in clinical trials as a methamphetamine abuse treatment. Lobeline interacts with nicotinic receptor subtypes, dopamine transporters (DATs), and vesicular monoamine transporters (VMAT2s). Methamphetamine inhibits VMAT2 and promotes dopamine (DA) release from syna...

Descripció completa

Guardat en:
Dades bibliogràfiques
Autors principals: Nickell, Justin R., Krishnamurthy, Sairam, Norrholm, Seth, Deaciuc, Gabriela, Siripurapu, Kiran B., Zheng, Guangrong, Crooks, Peter A., Dwoskin, Linda P.
Format: Artigo
Idioma:Inglês
Publicat: The American Society for Pharmacology and Experimental Therapeutics 2010
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC2812121/
https://ncbi.nlm.nih.gov/pubmed/19855096
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/jpet.109.160275
Etiquetes: Afegir etiqueta
Sense etiquetes, Sigues el primer a etiquetar aquest registre!