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Design and in vitro Characterization of Highly Sst(2)-selective Somatostatin Antagonists Suitable for Radio-Targeting

Radiolabeled sst(2) and sst(3) antagonists are better candidates for tumor targeting than agonists with comparable binding characteristics.1 Because the majority of neuroendocrine tumors express sst(2), we used the known antagonists Acetyl-pNO(2)Phe(2)-c[dCys(3)-Tyr(7)-dTrp(8)-Lys(9)-Thr(10)-Cys(14)...

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Autors principals: Cescato, Renzo, Erchegyi, Judith, Waser, Beatrice, Piccand, Véronique, Mäcke, Helmut R., Rivier, Jean E., Reubi, Jean Claude
Format: Artigo
Idioma:Inglês
Publicat: 2008
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC2789649/
https://ncbi.nlm.nih.gov/pubmed/18543899
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jm701618q
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