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Modifications at the C-Terminus to Improve Pyrrole-Imidazole Polyamide Activity in Cell Culture

Pyrrole-imidazole (Py-Im) hairpin polyamides are a class of small molecule DNA-minor groove binding compounds that have been shown to modulate endogenous gene expression in cell culture. Gene regulation by polyamides requires efficient cellular uptake and nuclear localization properties for candidat...

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Detalhes bibliográficos
Main Authors: Jacobs, Claire S., Dervan, Peter B.
Formato: Artigo
Idioma:Inglês
Publicado em: 2009
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC2788682/
https://ncbi.nlm.nih.gov/pubmed/19572551
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jm900256f
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