Substitution of Arginine with Proline and Proline Derivatives in Melanocyte-Stimulating Hormones Leads to Selectivity for Human Melanocortin 4 Receptor

Eitemau Tebyg

• Effects of Macrocycle Size and Rigidity on Melanocortin Receptor-1 and -5 Selectivity in Cyclic Lactam α-Melanocyte-Stimulating Hormone Analogs
  gan: Mayorov, Alexander V., et al.
  Cyhoeddwyd: (2006)
• Structure–activity studies of new melanocortin peptides containing an aromatic amino acid at the N-terminal position
  gan: Grieco, Paolo, et al.
  Cyhoeddwyd: (2005)
• Structure–Activity Relationships of Cyclic Lactam Analogues of α-Melanocyte-Stimulating Hormone (α-MSH) Targeting the Human Melanocortin-3 Receptor
  gan: Mayorov, Alexander V., et al.
  Cyhoeddwyd: (2007)
• Contribution of the Conserved Amino Acids of the Melanocortin-4 Receptor in D-[Nle(4),Phe(7)]-α-Melanocyte-stimulating Hormone Binding and Signaling(□S)
  gan: Chen, Min, et al.
  Cyhoeddwyd: (2007)
• Solid-Phase Peptide Head-to-Side Chain Cyclodimerization: Discovery of C(2)-Symmetric Cyclic Lactam Hybrid α-Melanocyte-Stimulating Hormone (MSH)/Agouti-Signaling Protein (ASIP) Analogues with Potent Activities at the Human Melanocortin Receptors
  gan: Mayorov, Alexander V., et al.
  Cyhoeddwyd: (2010)