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Substitution of Arginine with Proline and Proline Derivatives in Melanocyte-Stimulating Hormones Leads to Selectivity for Human Melanocortin 4 Receptor

A new series of melanotropin analogues with His or Arg residues in the core pharmacophores of MTII, SHU9119 and Ac-NDP-γ-MSH-NH(2) replaced by Pro or trans-/cis- 4-guanidinyl-Pro derivatives were designed and synthesized to introduce selectivity toward the human melanocortin 4 receptor (hMC4R). Anal...

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Detalhes bibliográficos
Main Authors: Qu, Hongchang, Cai, Minying, Mayorov, Alexander V., Grieco, Paolo, Zingsheim, Morgan, Hruby, Victor. J.
Formato: Artigo
Idioma:Inglês
Publicado em: 2009
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC2775485/
https://ncbi.nlm.nih.gov/pubmed/19473029
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jm801300c
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