Structure–Activity Relationships of Cyclic Lactam Analogues of α-Melanocyte-Stimulating Hormone (α-MSH) Targeting the Human Melanocortin-3 Receptor

A variety of dicarboxylic acid linkers introduced between the α-amino group of Pro(6) and the ε-amino group of Lys(10) of the cyclic lactam α-melanocyte-stimulating hormone (α-MSH)-derived Pro(6)-D-Phe7/D-Nal(2′)(7)-Arg(8)-Trp(9)-Lys(10)-NH(2) pentapeptide template lead to nanomolar range and select...

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Detalhes bibliográficos
Main Authors: Mayorov, Alexander V., Cai, Minying, Palmer, Erin S., Dedek, Matthew M., Cain, James P., Van Scoy, April R., Tan, Bahar, Vagner, Josef, Trivedi, Dev, Hruby, Victor J.
Formato: Artigo
Idioma:Inglês
Publicado em: 2007
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Article
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC2587288/
https://ncbi.nlm.nih.gov/pubmed/18088090
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jm070461w
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