Caricamento...

Cyclic Lactam Hybrid α-MSH/Agouti-Related Protein (AGRP) Analogues with Nanomolar Range Binding Affinities at the Human Melanocortin Receptors

A novel hybrid melanocortin pharmacophore was designed based on the topographical similarities between the pharmacophores of Agouti related protein (AGRP) an endogenous melanocortin antagonist, and α-melanocyte-stimulating hormone (α-MSH), an endogenous melanocortin agonist. When employed in two dif...

Descrizione completa

Salvato in:
Dettagli Bibliografici
Autori principali: Mayorov, Alexander V., Cai, Minying, Palmer, Erin S., Tanaka, Dustin K., Cain, James P., Dedek, Matthew M., Tan, Bahar, Trivedi, Dev, Hruby, Victor J.
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2011
Soggetti:
Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC3216836/
https://ncbi.nlm.nih.gov/pubmed/21486697
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmcl.2011.03.019
Tags: Aggiungi Tag
Nessun Tag, puoi essere il primo ad aggiungerne! !