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Zyklophin, a systemically active selective kappa opioid receptor peptide antagonist with short duration of action

The cyclic peptide zyklophin {[N-benzylTyr(1),cyclo(D-Asp(5),Dap(8))-dynorphin A-(1–11)NH(2), Patkar KA, et al. (2005) J Med Chem 48: 4500–4503} is a selective peptide kappa opioid receptor (KOR) antagonist that shows activity following systemic administration. Systemic (1–3 mg/kg s.c.) as well as c...

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Autors principals: Aldrich, Jane V., Patkar, Kshitij A., McLaughlin, Jay P.
Format: Artigo
Idioma:Inglês
Publicat: National Academy of Sciences 2009
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC2775281/
https://ncbi.nlm.nih.gov/pubmed/19841255
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1073/pnas.0910180106
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