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Novel Flufenamic Acid Analogs as Inhibitors of Androgen Receptor Mediated Transcription

The androgen receptor (AR), which mediates the signals of androgens, plays a crucial role in prostate related diseases. Although widely used, currently marketed anti-androgenic drugs have significant side effects. Several studies have revealed that non-steroidal anti-inflammatory drugs, like flufena...

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Hlavní autoři: Féau, Clémentine, Arnold, Leggy A., Kosinski, Aaron, Zhu, Fangyi, Connelly, Michele, Guy, R. Kiplin
Médium: Artigo
Jazyk:Inglês
Vydáno: 2009
Témata:
On-line přístup:https://ncbi.nlm.nih.gov/pmc/articles/PMC2763043/
https://ncbi.nlm.nih.gov/pubmed/19645433
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/cb900143a
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