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Structure-guided development of selective TbcatB inhibitors

The trypanosomal cathepsin TbcatB is essential for parasite survival and is an attractive therapeutic target. Herein we report the structure-guided development of TbcatB inhibitors with specificity relative to rhodesain and human cathepsins B and L. Inhibitors were tested for enzymatic activity, try...

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Autors principals: Mallari, Jeremy P., Shelat, Anang A., Kosinski, Aaron, Caffrey, Conor R., Connelly, Michele, Zhu, Fangyi, McKerrow, James H., Guy, R. Kiplin
Format: Artigo
Idioma:Inglês
Publicat: 2009
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC2762491/
https://ncbi.nlm.nih.gov/pubmed/19769357
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jm900908p
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